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YDL223C (HBT1) te kaihanga paura CAS No.: 489408-02-8 99% purea min.mo nga kai taapiri

Whakaahuatanga Poto:

Ko te HBT1 e herea ana ki te rohe here-ligand o te α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptor (AMPA-R) i roto i te glutamate-ti'aturi.


Taipitopito Hua

Tohu Hua

Tawhā Hua

ingoa hua

HBT1

Ko tetahi atu ingoa

YDL223C

CAS No.

489408-02-8

tātai rāpoi ngota

C16H17F3N4O2S

Te taumaha ngota

386.40

Maamaa

99.0%

Te ahua

Kowhai marama totoka

Te takai

1kg mo ia peeke 25kg mo ia pahu

Taupānga

nootropics

Whakataki hua

Ko te HBT1 e herea ana ki te rohe here-ligand o te α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptor (AMPA-R) i roto i te glutamate-ti'aturi.Ko te tikanga ko te HBT1 he ngota ngota ka taea anake te here ki nga waahi motuhake o te pūmua AMPA-R i te wa e noho ana te glutamate, a ka awhina tenei here ki te whakahaere i te mahi o te pūmua.Ko nga kaiwhakawhiwhi AMPA e whakaatuhia ana puta noa i te punaha nerve matua me te whai waahi nui ki te whakawhitiwhiti korero neuronal, te tukatuka tairongo, me te ako, te mahara, me te kirihou synaptic.Ko nga kaiwhakawhiwhi AMPA he kaikoha nui ki te neurotransmission whakahihiri, he takawaenga tere, he tere te whakaheke i te whakakorikori o te maha o nga synapses, ka uru ki nga urupare wawe o nga rohe synaptic ki te glutamate.Ko nga kaiwhakawhiwhi AMPA he maha nga wa e whakaatuhia ana me nga kaiwhakawhiwhi NMDA i nga synapses, me te whakatairanga tahi i nga tukanga kirihou synaptic e uru ana ki te ako, te mahara, te excitotoxicity, me te neuroprotection.

Āhuahira

Ko te tauwehe neurotrophic i ahu mai i te roro (BDNF) he mea neurotrophic e whai waahi nui ana ki te tiaki me te roha o nga neurons, a he kaha, he maha nga paanga ki te whakatipuranga, te rereketanga, te oranga me te mate o nga pūtau neuronal me te kore-neuronal, Acts as he neurotransmitter modulator me te whai wāhi ki te kirihou neuronal mo te ako me te mahara.Na reira he mea nui ki te hauora me te oranga o te punaha nerve.Ko te pikinga o te BDNF ka awhina i te maimoatanga me te aukati i nga tini mate.

Nga tono

Ko te HBT1 he pukapuka whakaihiihi kaikawe AMPA me te iti ake o te agonism ka whakaritea ki te LY451395 me OXP1, ka whakaawe i te hanga o te tauwehe neurotrophic i ahu mai i te roro (BDNF), a he iti nei te paanga ki nga neurons tuatahi Ko te Agitation.Ko te HBT1 e herea ana ki te rohe here-ligan o AMPA-R i roto i te ahua o te glutamate.Ka mahi tahi, ka whakatairanga i nga tukanga kirihou synaptic e uru ana ki te ako, te mahara, te hihiri me te neuroprotection.Ka taea te whakapai ake i te mohio me te mahara o te roro, me te whakarei ake i te kaha ako o te tangata.


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