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Kaihanga paura Nefiracetam Nama CAS: 77191-36-7 99% te parakore iti rawa mō ngā kai tāpiringa

Whakaahuatanga Poto:

Kei roto te Nefiracetam i te akomanga rongoā whakarei ake i te hinengaro kāore i te rohe, he rerekē ngā hanganga matū o ēnei, ā, ka whakarei ake i te kaha hinengaro me te ārai i te kino o te ako me te mahara mā ō rātou pānga ki te roro.


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Ataata Hua

Ngā Tawhā Hua

Ingoa hua

Nefiracetam

Ingoa kē atu

n-(2,6-dimethylphenyl)-2-oxo-1-pyrrolidineacetamide;NEFIRACETAM;

2-oxo-1-pyrrolidinylaceticacid,2,6-dimethylanilide;

dm9384;

n-(2,6-dimethylphenyl)-2-oxo-1-pyrrolidineacetamid;DM-9384,(2-(2-Oxopyrrolidin-1-yl)-N-(2,6-dimethylphenyl)-acetamide);

DMMPA

Nama CAS

77191-36-7

Tātai ngota

C14H18N2O2

Taumaha ngota

246.3

Te parakore

99.0%

Āhua

Paura mā

Te tākai

25 kg/peera

Tono

nootropic

Whakataki hua

Nō te whānau piracetam te Nefiracetam, he momo rongoā e mōhiotia ana mō ōna āhuatanga whakarei ake i te hinengaro. I hangaia tuatahitia a Nefiracetam i te tīmatanga o te tekau tau atu i 1980, ā, i tere te aro atu nā tōna tikanga mahi ahurei me ngā whakamahinga rongoā pea. E whakaarohia ana ka pā tēnei matū racemic ki ngā neurotransmitters me ngā kaiwhakawhiwhi i roto i te roro, ā, ka whakatairanga i te whakapai ake i ngā pūkenga hinengaro. Ko te Nefiracetam te mea nui ki ngā taumata o te acetylcholine i roto i te roro, he neurotransmitter matua e kawenga ana mō te mahara, te ako, me te mahi hinengaro. Mā te whakarerekē i ngā kaiwhakawhiwhi acetylcholine, ka whakatairanga te nefiracetam i te whakapiki i te whakawhitiwhiti kōrero i waenga i ngā neurons, ā, ka whakarei ake i te kirihou synaptic me te whakapai ake i te pupuri mahara. Hei tāpiri, ka taunekeneke te nefiracetam me ngā kaiwhakawhiwhi waikawa gamma-aminobutyric (GABA) hei āwhina i te taurite i te taiao neurotransmitter. Mā te pānga pai ki ngā neurotransmitters whakaoho me te aukati, ka āwhina te nefiracetam ki te pupuri i te mahi pai o te roro, ā, ka whakapai ake i te arotahi, te aro, me te mahi hinengaro whānui.

Āhuatanga

(1) Teitei o te parakore: Ka taea e Nefiracetam te whiwhi hua tino parakore mā te whakamahine i ngā tukanga whakaputa. Ko te tikanga o te tino parakore he pai ake te wātea o te koiora me te iti ake o ngā urupare kino.

(2) Haumarutanga: He tino haumaru, he iti noa ngā pānga kino.

(3) Te Pūmautanga: He pai te pumau o Nefiracetam, ā, ka taea e ia te pupuri i tōna mahi me tōna pānga i raro i ngā taiao me ngā tikanga rokiroki rerekē.

Ngā tono

Ko te Nefiracetam he matū hydrophobic o te piracetam, e kiia whānuitia ana ko te matū e whai kawenga ana mō te kitenga o ngā hongere konupūmā i roto i te tinana me te whakawhiti ā-kore o ngā matū tohu whakaoho hei agonist wāhanga o ngā hongere ion konupūmā. Te pae here glycine o te kaiwhakawhiwhi NDMA. Mā tōna pānga ki te cortex roro, ka taea e te nefiracetam te whakarei ake i ngā pūkenga hinengaro me te ārai i te ngoikore o te ako me te mahara. Kāore he āhuatanga agonist receptor muscarinic, he āhuatanga antagonist rānei, kāore hoki e aukati i te mahi acetylcholinease. Nō reira, ko ōna pānga anti-amnestic me te whakarei ake i te mahara ka tutuki mā te whakapai ake i te tukunga o te acetylcholine i roto i te cortex roro.


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