Nefiracetam paura kaihanga CAS Nama: 77191-36-7 99% purea min.mo nga kai taapiri
Tawhā Hua
| ingoa hua | Nefiracetam |
| Ko tetahi atu ingoa | n-(2,6-dimethylphenyl)-2-oxo-1-pyrrolidineacetamide;NEFIRACETAM; 2-oxo-1-pyrrolidinylaceticacid,2,6-dimethylanilide; dm9384; n-(2,6-dimethylphenyl)-2-oxo-1-pyrrolidineacetamid;DM-9384,(2-(2-Oxopyrrolidin-1-yl) -N-(2,6-dimethylphenyl)-acetamide); DMMPA |
| CAS No. | 77191-36-7 |
| tātai rāpoi ngota | C14H18N2O2 |
| Te taumaha ngota | 246.3 |
| Maamaa | 99.0% |
| Te ahua | Te paura ma |
| Te takai | 25 kg/paera |
| Taupānga | nootropic |
Whakataki hua
No roto a Nefiracetam i te karaehe o nga raau taero e whakanui ana i te matauranga kore-rohe, he rereke nga hanganga matū me te whakarei ake i te kaha o te hinengaro me te aukati i te kino o te ako me te mahara ma o raatau paanga ki te uho roro.Kaore he ahuatanga o nga agonists receptor muscarinic me nga antagonists, kaore hoki e aukati i te mahi a Ach.Ko nga hua anti-wareware me te whakanui i te mahara o tenei tarukino ka tutuki ma te whakarei ake i te tukunga o Ach i roto i te uho roro.Ko nga kinases pūmua e whakawhirinaki ana ki te puni ka whakarei ake i te mahi hongere Ca2+, tera pea te haepapa mo to raatau tukunga Ach.Ko te Nefiracetam (NEF) he kaihoko nootropic momo pyrrolidone me nga momo rongoa rongoa tae atu ki nga paanga whakarei ake.I roto i nga mate o te amygdala, ka whakakorehia e te nefiracetam nga hopukanga electroencephalographic me te whanonga.Kei a NEF tetahi awhi anticonvulsant motuhake.
Āhuahira
Ka whakamahia te Nefiracetam ki te rongoa i nga mate pukupuku.Ka taea e ia te whakarei ake i te kaha o te hinengaro me te aukati i te kino o te ako me te mahara na tona paanga ki te uho roro.Kaore he ahuatanga o te agonist receptor muscarinic me te kaihoko antagonistic, kaore hoki e aukati i te mahi a te acetyl cholinase.Na reira, ka puta mai ona paanga anti-wareware me te whakanui ake i te mahara ma te whakapai ake i te tukunga o te acetylcholine i roto i te cortex cerebral.
Nga tono
Ko te Nefiracetam he pärönaki hydrophobic o te piracetam me te whakahiatotanga waihanga o nga puhui Racetam katoa piracetam.Ko te Nefiracetam i hangaia e Daiichi Sankyo (kamupene rongoa Japanese) mo te maimoatanga o AD.I tua atu i nga tikanga katoa e kii ana ki a Nefiracetam, i te nuinga o te waa ka whakaarohia he matū te kawenga mo te kitenga o nga awa konupūmā i roto i te tinana, me te whakawhitinga autaki o te matū tohu whakaihiihi, e mahi ana hei agonist waahanga o te pae here-glycine o te kaiutuutu NDMA.
