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Kaihanga paura matū 7P Nama CAS: 1890208-58-8 99% te parakore iti rawa mō ngā kai tāpiringa

Whakaahuatanga Poto:

I whakaaturia te kaha o te matū 7p ki te whakaoho i te tipu o ngā axon GAP-43-pai i roto i tētahi tauira kararehe o te whara o te io whatu, e whakaatu ana ko te mahi tipu neurite o te matū 7p i roto i te vitro ka puta he whakaoho i te whakaoranga axon i roto i te tinana ora.


Taipitopito Hua

Ngā Tohu Hua

Ataata Hua

Ngā Tawhā Hua

Ingoa hua

Pūhui 7P

Ingoa kē atu

Pūhui7P;2-[(2-methoxyphenyl)[(4-methylphenyl)sulfonyl]amino]-N-(4-methoxy-3-pyridinyl)acetamide;

2-(N-(2-methoxyphenyl)-4-methylphenylsulfonamido)-N-(4-methoxypyridin-3-yl)acetamide

Nama CAS

1890208-58-8

Tātai ngota

C22H23N3O5S

Taumaha ngota

441.51

Te parakore

99.0%

Āhua

Paura mā

Tono

Nootropic

Whakataki hua

Ko te matū 7P e pā ana ki tētahi matū waro motuhake kei roto e whitu ngā ngota waro. I roto i te matū waro, he huānga nui te waro nā te mea ka taea e ia te hanga hononga pumau me ētahi atu ngota, tae atu ki ngā ngota waro, hei hanga i ngā ngota matatini. He maha ngā āhuatanga me ngā mahi a ēnei ngota, ka waiho ngā matū waro hei poraka hanga o te ora. I roto i ngā tauira kararehe o te whara o te io whatu, i whakaaturia te matū 7p ki te whakaoho i te tipu o ngā axon GAP-43-pai, e kī ana ko te mahi tipu neurite o te matū 7p i roto i te vitro ka huri hei whakaoho i te whakahoutanga axonal i roto i te vivo. Ko te paura matū 7P he paura ma ki te ma-pango i hangaia hei matū takirua mō te tautuhi i ngā aukati aukati thromboxane receptor takirua. Inaa, i whakaatu te matū 7p i te whiriwhiringa mō te prostaglandin I2 synthase (PTGIS, CYP8A1) e pā ana ki te thromboxane synthase (CYP5A1). Ka whakatairanga te paura matū nootropic 7P i te tipu o ngā axon Gap-43-pai, ā, ka whakaoho i te whakahoutanga axonal i roto i te tinana. Kua hangaia te Matatini 7p kounga teitei hei whakapai ake i te taunga, hei whakapai ake i te wairua, hei āwhina hoki ki te whawhai ki te ngenge. Ka ārai hoki i te waikura o te roro, ā, ka āwhina hoki ki te whawhai ki ngā kino o te roro i puta mai i te inu waipiro.

Āhuatanga

结构图

(1) Teitei o te parakore: Ka taea e te matū 7P te whiwhi hua tino parakore mā roto i ngā tukanga whakaputa kua whakatikatikaina. Ko te tikanga o te tino parakore he pai ake te wātea o te koiora me te iti ake o ngā tauhohenga kino.

(2) Haumaru: Kua whakamātauhia te haumaru o te matū 7P mō te tinana tangata.

(3) Te Pūmautanga: He pai te pumau o te matū 7P, ā, ka taea e ia te pupuri i tōna kaha me tōna pānga i raro i ngā taiao me ngā tikanga rokiroki rerekē.

Ngā tono

Ka whakarei ake te matū 7p i te tipu o ngā neuron tuatahi kua whakatipuria mai i te hippocampus, te cortex roro, me te retina, ā, ka whakaoho i te whakahoutanga o te io whatu i roto i ngā tauira kararehe o te whara o te io whatu. Ka whakarei ake hoki i te mahi tahi, ka rongoā i te kino o te roro e pā ana ki te waipiro, ā, ka ārai i te waikura huri noa i te roro. Ka āwhina hoki ki te whakapai ake i te wairua me te whawhai ki te ngenge.


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